生物活性:3-Hydroxy agomelatine-d3 is a deuterium labeled 3-Hydroxy agomelatine. 3-Hydroxy agomelatine is a 5-HT2C receptor antagonist with an IC50 of 3.2 μM and a Ki of 1.8 μM[1].
IC50 & Target[1]:5-HT2C Receptor
3.2 μM (IC50)
5-HT2C Receptor
1.8 μM (Ki)
分子量:262.32
Formula:C15H14D3NO3
CAS 号:1079774-23-4
非标记 CAS:166526-99-4
性状:固体
颜色:Off-white to light yellow
中文名称:3-羟基阿戈美拉汀杂质7-d3
运输条件:Room temperature in continental US; may vary elsewhere.
储存方式:Powder:-20°C:3 years,4°C:2 years
In solvent:-80°C:6 months,-20°C:1 month