生物活性:Navitoclax-d8 is the deuterium labeled Navitoclax. Navitoclax (ABT-263) is a potent and orally active Bcl-2 family protein inhibitor that binds to multiple anti-apoptotic Bcl-2 family proteins, such as Bcl-xL, Bcl-2 and Bcl-w, with a Ki of less than 1 nM[1].
体外研究(In Vitro):氢、碳和其他元素的稳定重同位素已被掺入药物分子中,主要用作药物开发过程中定量的示踪剂。氘代因其可能影响药物的药代动力学和代谢特征而受到关注[1]。
瑞禧生物 has not independently confirmed the accuracy of these methods. They are for reference only.
Navitoclax-d8 相关抗体:
Bcl-2 Antibody
Bcl2 Antibody
Bax Antibody (YA591)
Bad Antibody
Bak Antibody (YA592)
BAX Antibody (YA825)
Bcl-XL Antibody
Bim Antibody
BNIP3 Antibody
PUMA Antibody
MCL1 Antibody
Bak Antibody
Bax Antibody (YA826)
Bcl2 Antibody (YA824)
BNIP3L Antibody
BAG2 Antibody (YA1398)
Phospho-PML Protein (Ser518) Antibody (YA2632)
Bid Antibody
BAG1 Antibody (YA932)
BAG1 Antibody (YA933)
Bcl10 Antibody (YA1188)
BAP31 Antibody (YA1320)
BCL2L1 Antibody (YA1359)
BAG3 Antibody (YA2240)
Bok Antibody (YA2289)
BPR Antibody (YA2393)
DYNLL1 Antibody (YA2724)
Bcl2 L14 Antibody (YA2740)
Bcl2 A1 Antibody (YA2743)
Phospho-Bad (Ser112) Antibody (YA3099)
分子量:982.66
Formula:C47H47D8ClF3N5O6S3
CAS 号:1217620-38-6
非标记 CAS:923564-51-6
性状:固体
颜色:White to off-white
中文名称:生根粉263 d8
运输条件:Room temperature in continental US; may vary elsewhere.
储存方式:Powder:-20°C:3 years
In solvent:-80°C:6 months,-20°C:1 month