生物活性：Cariprazine-d6 is a deuterium labeled Cariprazine. Cariprazine Cariprazine is an antipsychotic agent that exhibits high affinity for the D3 (Ki of 0.085 nM) and D2 (Ki of 0.49 nM) receptors, and moderate affinity for the 5-HT1A receptor (Ki of 2.6 nM)[1].
IC50 & Target[1]：Dopamine D2 Receptor
0.49 nM (Ki)
Dopamine D3 Receptor
0.085 nM (Ki)
5-HT1A Receptor
2.6 nM (Ki)
分子量：433.45
Formula：C21H26D6Cl2N4O
CAS 号：1308278-67-2
非标记 CAS：839712-12-8
性状：固体
颜色：White to off-white
中文名称：卡利拉嗪 d6
运输条件：Room temperature in continental US; may vary elsewhere.
储存方式：Powder：-20°C：3 years，4°C：2 years
In solvent：-80°C：6 months，-20°C：1 month