生物活性:Gefitinib-d8 is a deuterium labeled Gefitinib. Gefitinib is an EGFR tyrosine kinase inhibitor, with IC50 of 2-37 nM in NR6wtEGFR cells[1][2].
IC50 & Target:IC50: 37 nM (Tyr1173 site, in NR6wtEGFR cells), 37 nM (Tyr992 site, in NR6wtEGFR cells)[1]
分子量:454.95
Formula:C22H16D8ClFN4O3
CAS 号:857091-32-8
非标记 CAS:184475-35-2
性状:固体
颜色:White to off-white
中文名称:吉非替尼 d8
运输条件:Room temperature in continental US; may vary elsewhere.
储存方式:Powder:-20°C:3 years,4°C:2 years
In solvent:-80°C:6 months,-20°C:1 month